|
Mutation Information
|
Mutation Site
|
V82F |
|
Mutation Type
|
Amino acid level |
|
Gene/Protein/Region Type
|
RT |
|
Relevant Drug
|
nevirapine (NPV) |
Literature Information
|
PubMed PMID
|
32140396
|
|
Published Year
|
2020 |
|
Journal
|
Acta pharmaceutica Sinica. B |
|
Title
|
Synthesis and biological evaluation of a series of 2-(((5-akly/aryl-1H-pyrazol-3-yl)methyl)thio)-5-alkyl-6-(cyclohexylmethyl)-pyrimidin-4(3H)-ones as potential HIV-1 inhibitors. |
|
Author
|
Wu Y,Tang C,Rui R,Yang L,Ding W,Wang J,Li Y,Lai CC,Wang Y,Luo R,Xiao W,Zhang H,Zheng Y,He Y |
|
Evidence
|
Table 2
|
|
|