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Basic Characteristics of Mutations
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Mutation Site
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H275Y |
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Mutation Site Sentence
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These data demonstrate that despite an increase in H275Y variants in 2011, there was no marked change in the frequency of peramivir- or laninamivir-resistant variants following the market release of the drugs in Japan in 2010. |
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Mutation Level
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Amino acid level |
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Mutation Type
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Nonsynonymous substitution |
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Gene/Protein/Region
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NA |
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Standardized Encoding Gene
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NA
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Genotype/Subtype
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H1N1 |
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Viral Reference
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-
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Functional Impact and Mechanisms
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Disease
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Influenza A
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Immune
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- |
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Target Gene
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-
|
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Clinical and Epidemiological Correlations
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Clinical Information
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- |
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Treatment
|
- |
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Location
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Australia; Brunei; Cambodia; Fiji; Hong Kong; Kenya; Macau (SAR; China); Malaysia; New Caledonia; New Zealand; Papua New Guinea; Philippines; Singapore; Solomon Islands; South Africa; South Korea; Sri Lanka; Taiwan; Thailand |
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Literature Information
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PMID
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24734292
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Title
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Peramivir and laninamivir susceptibility of circulating influenza A and B viruses
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Author
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Leang SK,Kwok S,Sullivan SG,Maurer-Stroh S,Kelso A,Barr IG,Hurt AC
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Journal
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Influenza and other respiratory viruses
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Journal Info
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2014 Mar;8(2):135-9
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Abstract
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Influenza viruses collected from regions of Asia, Africa and Oceania between 2009 and 2012 were tested for their susceptibility to two new neuraminidase inhibitors, peramivir and laninamivir. All viruses tested had normal laninamivir inhibition. However, 3.2% (19/599) of A(H1N1)pdm09 viruses had highly reduced peramivir inhibition (due to H275Y NA mutation) and <1% (6/1238) of influenza B viruses had reduced or highly reduced peramivir inhibition, with single occurrence of variants containing I221T, A245T, K360E, A395E, D432G and a combined G145R+Y142H mutation. These data demonstrate that despite an increase in H275Y variants in 2011, there was no marked change in the frequency of peramivir- or laninamivir-resistant variants following the market release of the drugs in Japan in 2010.
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Sequence Data
|
-
|