|
Basic Characteristics of Mutations
|
|
Mutation Site
|
K65R |
|
Mutation Site Sentence
|
Higher rates of NRTI, NNRTI, K65R tenofovir resistance, and multi-class resistance were found compared to those reported in literature. |
|
Mutation Level
|
Amino acid level |
|
Mutation Type
|
Nonsynonymous substitution |
|
Gene/Protein/Region
|
RT |
|
Standardized Encoding Gene
|
gag-pol:155348
|
|
Genotype/Subtype
|
HIV-1 CRF01_AE |
|
Viral Reference
|
-
|
|
Functional Impact and Mechanisms
|
|
Disease
|
HIV Infections
|
|
Immune
|
- |
|
Target Gene
|
-
|
|
Clinical and Epidemiological Correlations
|
|
Clinical Information
|
Y |
|
Treatment
|
tenofovir (TDF) |
|
Location
|
Philippines |
|
Literature Information
|
|
PMID
|
32081778
|
|
Title
|
High rates of tenofovir failure in a CRF01_AE-predominant HIV epidemic in the Philippines
|
|
Author
|
Salvana EMT,Samonte GMJ,Telan E,Leyritana K,Tactacan-Abrenica RJ,Ching PR,Arevalo GM,Dungca NT,Penalosa-Ramos C,Mendoza KAR,Trinidad LF,Tonga AD,Lim J,Destura R,Alejandria M,Solante R,Arcangel L,Palaypayon NS,Schwem BE
|
|
Journal
|
International journal of infectious diseases : IJID : official publication of the International Society for Infectious Diseases
|
|
Journal Info
|
2020 Jun;95:125-132
|
|
Abstract
|
BACKGROUND: The Philippines has the fastest growing HIV epidemic in the Asia-Pacific. This increase was accompanied by a shift in the predominant HIV subtype from B to CRF01_AE. Increasing evidence points to a difference in treatment responses between subtypes. We examined treatment failure and acquired drug resistance (ADR) in people living with HIV (PLHIVs) after one year on antiretrovirals (ARVs). METHODS: PLHIV maintained on ARVs for one year were recruited. Treatment failure was defined as a viral load of >/=1000 copies/mL. Sanger sequencing for genotyping and drug resistance mutation (DRM) detection was performed on patients failing treatment. RESULTS: 513 PLHIV were enrolled. The most common antiretroviral regimens were TDF+3TC + EFV (269) and AZT+3TC + EFV (155). 53 (10.3%) subjects failed treatment. Among these, 48 (90.6%) had DRMs, 84.9% were subtype CRF01_AE. Tenofovir-based regimens performed worse than zidovudine-based regimens (OR 3.28, 95% CI 1.58-7.52 p < 0.001). Higher rates of NRTI, NNRTI, K65R tenofovir resistance, and multi-class resistance were found compared to those reported in literature. CONCLUSIONS: HIV treatment failure at one year of treatment in the Philippines is 10.3%. We found unusually high tenofovir and multiclass resistance, and optimal ARV regimens may need to be reevaluated for CRF01_AE-predominant epidemics.
|
|
Sequence Data
|
-
|
|
|